Drug Database
TE

testosterone enanthate (Vibex QS T / QS T / Xyosted)

✓ Approved

Antares Pharma, Inc. · AR · 类固醇

什么是 testosterone enanthate?

testosterone enanthate 是一种类固醇,由Antares Pharma, Inc.研发。该药已获批,用于治疗相关适应症,给药途径:Injectable (Others)、Subcutaneous Injection。

药物档案

商品名Vibex QS T, QS T, Xyosted
公司Antares Pharma, Inc.
药物类别类固醇, 小分子
分子靶点AR
给药途径Injectable (Others), Subcutaneous Injection
状态Approved

作用机制

分子靶点

testosterone enanthate 作用于 1 个分子靶点:

ARandrogen receptor (DHTR, AR8)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

testosterone enanthate 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Endocrine disordersHypogonadism✓ Approved

相关研究文献

PubMedAmerican journal of physiology. Lung cellular and molecular physiology2026-08-05

Testosterone alleviates inflammation but increases the methacholine response in male mice with allergic lung inflammation.

Henry Cyndi C, Boucher Magali M, Rojas-Ruiz Andrés A, Camillari Louane L et al.

Testosterone seems protective against asthma, but the underlying mechanisms are uncertain. Although several of its anti-inflammatory properties have been described, its effect on respiratory mechanics and the methacholine response are incompletely understood. Herein, the effect of testosterone was investigated on several features of experimental asthma with a special focus on respiratory mechanics and the methacholine response. Systemic testosterone was first altered to subphysiological, physiological, or supraphysiological levels in male BALB/c mice through orchiectomy and testosterone supplementation. Testosterone (0.25 mg/day/30 g of body weight) was delivered continuously during 20 days using an implanted pump. At day 10, each group was exposed intranasally to either saline or house dust mite (HDM) once-daily for 10 consecutive days to induce allergic lung inflammation. The day after the last exposure, respiratory mechanics were measured at baseline and in response to nebulized methacholine. Bronchoalveolar lavages (BAL) and lung tissues were also collected to quantify inflammation. Baseline respiratory mechanics were altered in mice with subphysiological levels of testosterone, with signs of small airway narrowing heterogeneity and closure. Testosterone drastically inhibited the HDM-induced inflammation. Yet, testosterone also increased the methacholine response, which occurred to the same extent in mice with and without experimental asthma. It is concluded that testosterone improves baseline respiratory mechanics and, although it increases the methacholine response, it does not synergistically amplify hyperresponsiveness in a context of experimental asthma probably because it concurrently decreases inflammation.

PMID 42552756
阅读全文 →
PubMedReproductive sciences (Thousand Oaks, Calif.)2026-08-05

Accurate Measurement of Serum Free Testosterone Levels via Liquid Chromatography‒Tandem Mass Spectrometry (LC‒MS/MS) has Predictive Value in the Diagnosis of Polycystic Ovary Syndrome and Associated Metabolic Disorders.

Liu Yang Y, Li Cheng C, Li Jie J, Wei Zhaolian Z et al.

Polycystic ovary syndrome (PCOS), in which hyperandrogenism is a major feature, is the most prevalent endocrine disorder among women of reproductive age. Serum free testosterone (FT) reflects the biologically active fraction of circulating testosterone. Accurate assessment of FT allows for precise identification of hyperandrogenism and provides critical guidance for the diagnosis of PCOS. Women with PCOS and normal controls (NCs) were included in this study. Fasting serum samples were collected during the early follicular phase to evaluate key clinical parameters, and FT levels were quantified using liquid chromatography‒tandem mass spectrometry (LC‒MS/MS). The diagnostic value of FT for identifying PCOS was assessed using Spearman's correlation analysis and receiver operating characteristic curves. A total of 202 women were included in the PCOS group, 121 were included in the NC group. Total testosterone (TT), free androgen index (FAI), and FT levels were significantly greater in the PCOS group than in the NC group. Both FAI and FT were positively correlated with body mass index (BMI), triglycerides, low-density lipoprotein cholesterol, fasting insulin and the homeostasis model assessment for insulin resistance; and were negatively correlated with high-density lipoprotein cholesterol. Following age and BMI adjustments, the area under the curve (AUC) for FT (AUC = 0.886) was greater than that for TT (AUC = 0.856) or FAI (AUC = 0.864). Compared with conventional assessments of TT and FAI, LC-MS/MS-based measurements of FT demonstrate superior diagnostic performance for identifying PCOS. Both FT and FAI are associated with obesity and the features of metabolic syndrome in PCOS patients.

PMID 42552471
阅读全文 →
PubMedFrontiers in physiology2026-08-05

Multimodal indicators of non-functional overreaching in NCAA Division I American football athletes: evidence for role-specific physiological adaptation.

Aychman Mackenzie M MM, Vinson Kelsey K, Tasnim Noor N, Perez Jorge J et al.

The purpose of this study was to characterize longitudinal patterns associated with non-functional overreaching (NFOR) in NCAA Division I American football athletes across a competitive season using salivary biomarkers, neuromuscular performance measures, and recovery metrics, with exploratory analyses by team role. Thirty-nine male athletes (age 20.4 ± 1.75 years) were monitored across a 15-week competitive season. Saliva samples collected pre-, mid-, and post-season assessed cortisol, testosterone, interleukin-6 (IL-6), and tumor necrosis factor-alpha (TNF-α). Neuromuscular performance was evaluated using countermovement jump metrics (jump height, normalized peak power and force, reactive strength index-modified [RSImod]) and PlayerLoad, while recovery was tracked via twice-weekly self-reports of sleep quality and muscle soreness. Associations among biomarkers, recovery, and performance were examined by starting status and position group; statistical significance was set at p ≤ 0.05. Distinct role-dependent patterns emerged. Among starters, higher testosterone-to-cortisol ratios were associated with lower soreness and better sleep quality, while higher IL-6/cortisol ratios were associated with higher RSImod values. Non-starters showed patterns consistent with greater physiological strain, with higher IL-6/cortisol ratios associated with poorer recovery despite lower external loads. Mid-season declines in countermovement jump performance coincided with biomarker changes suggestive of accumulated fatigue. Overall, both starters and non-starters exhibited patterns consistent with NFOR, though physiological signatures differed by role. Salivary biomarker ratios, particularly IL-6/cortisol, alongside neuromuscular measures such as RSImod may provide useful, non-invasive indicators of fatigue-related stress and support role-specific recovery strategies in applied sport settings.

PMID 42553027
阅读全文 →
PubMedNature reviews. Urology2026-08-04

Routine testosterone screening in military personnel: an opportunity for evidence-based implementation in men's health.

Mubarak Mohamed M, Modgil Vaibhav V

PMID 42547845
阅读全文 →
PubMedEuropean journal of endocrinology2026-08-04

Chronic Subcutaneous Kisspeptin-10 Stimulates Gonadotropin Secretion for 12 Days in Healthy Men.

Yeung Arthur C AC, Phylactou Maria M, Koysombat Kanyada K, Tsoutsouki Jovanna J et al.

To develop a protocol for chronic kisspeptin administration that persistently stimulates gonadotropin secretion. We evaluated the effects of acute and chronic subcutaneous kisspeptin-10 administration on reproductive hormones in healthy men to: (i) characterize the acute dose-response relationship to subcutaneous kisspeptin-10 infusion, (ii) assess the effects of continuous kisspeptin-10 infusion over 5-days, (iii) daily intermittent administration (8-hours on, 16-hours off) for 12-days. Randomized, single-blinded, placebo-controlled study. Overall, 15 healthy men were recruited (Study 1: n=7, Study 2: n=4; Study 3: n=7); 12 men served as controls. Luteinizing hormone (LH), follicle stimulating hormone (FSH) and testosterone, were assessed during an acute 8-hour dose-response subcutaneous kisspeptin-10 infusions (1.25-10.0 nmol/kg/h). Thereafter, we evaluated chronic subcutaneous administration, including continuous kisspeptin-10 infusion at 180 nmol/h for 5-days, and daily 8-hour infusions at 150 nmol/h for 12-days. (i) Acute subcutaneous kisspeptin-10 infusions dose-dependently increased LH, FSH, and testosterone vs vehicle (p<0.0001). (ii) Although testosterone concentrations remained elevated after 5-days of continuous kisspeptin-10, gonadotropin concentrations were similar to vehicle. (iii) Daily 8h subcutaneous infusions over 12-days sustained increases in gonadotropins (mean LH increase: vehicle -0.16 ±0.19; Day 1: +1.68 ±0.25; Day 12: +1.14 ±0.33, p=0.003 vs vehicle). Following 12-days, gonadotropin rises were still detected after kisspeptin-10 bolus (1nmol/kg) indicating that the kisspeptin receptor remained functional. We demonstrate that chronic subcutaneous kisspeptin administration sustain gonadotropin and testosterone secretion in healthy men for 12-days. These data can inform development of chronic kisspeptin administration protocols for the treatment of reproductive disorders.

PMID 42549827
阅读全文 →
PubMedJournal of pediatric surgery2026-08-04

Gonadal function and fertility outcomes after orchiopexy versus orchiectomy for testicular torsion: a systematic review and meta-analysis.

Nasr Aya M AM, Zamlout Ali A, Alghzawi Hamzah M HM, Youssef Youssef Ali YA et al.

To review the early and late changes in hormonal profiles, semen parameters, and clinical outcomes in patients treated with orchiopexy versus orchiectomy for testicular torsion. A systematic search was conducted across MEDLINE, Scopus, Web of Science, Cochrane Library, and other databases, following PRISMA guidelines. FSH, LH, testosterone, inhibin-B, and semen parameters. Quality was assessed using the Newcastle-Ottawa Scale. Certainty of evidence was evaluated using the GRADE framework. Statistical analysis was performed using the random-effects model. Eleven studies involving 538 participants (197 orchiectomy, 341 orchiopexy) were included. Orchiectomy was associated with a significant increase in FSH (SMD: 1.63, P<0.0001) and LH (SMD: 1.31, P<0.0001) compared to orchiopexy. However, testosterone (MD: 0.31 ng/mL; P=0.4) and inhibin-B (SMD: -0.14; P=0.87) levels were comparable between groups. Regarding semen parameters, orchiectomy resulted in a significant reduction in sperm concentration (MD: -18 million/mL, P=0.01). No significant differences were found in sperm count (MD: 13.9 million; P=0.43), normal morphology (MD: 4.97%; P=0.12), or total motility (MD: 4.05%; P=0.49). The pooled rate for ipsilateral atrophy following orchiopexy was 38%, which likely depends on ischemia duration. Surgical choice in testicular torsion does not significantly affect the overall hormonal balance or most semen parameters due to compensatory mechanisms of the hypothalamic-pituitary-gonadal axis. Clinical decisions should consider individual case factors, as we lack reliable data on subsequent paternity rates.

PMID 42546903
阅读全文 →

注册免费账户还可查看另外 9996 篇文献

免费注册查看全部文献 →

了解更多testosterone enanthate