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urea (Emolienta / urea, Vinas)

✓ Approved

Vinas · 小分子 · 小分子

什么是 urea?

urea 是一种小分子,由Vinas研发。该药已获批,用于治疗相关适应症,给药途径:Topical。

药物档案

商品名Emolienta, urea, Vinas
公司Vinas
药物类别小分子
给药途径Topical
状态Approved

治疗适应症

urea 针对 4 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Skin and subcutaneous tissue disordersDermatitis allergic✓ Approved
Skin and subcutaneous tissue disordersDermatitis atopic✓ Approved
Skin and subcutaneous tissue disordersDermatitis contact✓ Approved
Skin and subcutaneous tissue disordersPsoriasis✓ Approved

相关研究文献

PubMedBMC neurology2026-06-13

Ammonia storm: unmasking a suspected rare proximal urea cycle disorder in adulthood.

Vikhe Vikram V, Shaik Md Hassan MH, Khaire Priya P, Patil Rahul R et al.

Hyperammonaemia is a medical emergency which is mostly associated with liver dysfunction. However, in the absence of hepatic disease, rare inborn errors of metabolism such as urea cycle disorders (UCDs) must be considered. While UCDs typically present in the neonatal period, partial enzyme deficiencies may remain clinically silent until adulthood and present abruptly with life-threatening hyperammonaemia encephalopathy. Among these, late-onset carbamoyl phosphate synthetase I (CPS-I) deficiency is exceedingly rare and often underdiagnosed. We report a 32-year-old male who presented with acute onset altered sensorium progressing to coma over 12 h. The neurological decline was preceded by two to three episodes of vomiting on the day of admission and a recent history of a five-to-six-day febrile illness accompanied by gastrointestinal symptoms. On admission, the patient had a Glasgow Coma Scale score of 7/15 and required endotracheal intubation with ventilatory support. Routine laboratory investigations, including liver and renal function tests, were within normal limits. Neuroimaging studies (CT and MRI brain) showed no abnormalities. Plasma ammonia was markedly elevated at 397 µg/dL (Normal: <50 µg/dL), which rapidly escalated to 804 µg/dL within 24 h despite initial pharmacological intervention. Further metabolic evaluation revealed low plasma citrulline, elevated glutamine levels, and low urinary orotic acid, suggestive of a proximal urea cycle defect such as carbamoyl phosphate synthetase I (CPS-I) or N-acetylglutamate synthase (NAGS) deficiency. A significant family history of consanguinity and unexplained neonatal death, further supported a genetic etiology. The patient underwent urgent haemodialysis for ammonia clearance and was treated with protein restriction, dextrose-based intravenous fluids, and ammonia-lowering agents including sodium benzoate. His neurological status improved progressively, allowing successful extubation after three days. He was later discharged on oral L-citrulline supplementation and dietary protein restriction. At two-week follow-up, he was clinically stable with normalized plasma ammonia levels. This case highlights the importance of considering late-onset urea cycle disorders in adults presenting with unexplained hyperammonaemia encephalopathy. Early recognition and prompt aggressive management can be lifesaving and lead to complete neurological recovery.

PMID 42286544
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PubMedJournal of dairy science2026-06-13

The effect of the type of protein supplementation on splanchnic and mammary metabolism of dairy cows fed grass silage-based diets.

Roy C C, Ouellet D R DR, Pellerin D D, Lapierre H H

The current experiment studied 2 situations proposed to lead to decreased milk protein yield (MPY). First, NRC (2001) predicts that substitution of soybean meal (SBM) by canola meal (CM) decreases MP supply, thereby negatively affecting MPY. Second, excess RDP supply has a negative effect on post-liver AA supply, and hence, on MPY. These 2 potentially negative situations were tested through 1) substitution of SBM by CM in a grass-silage based diet, and 2) with an excess RDP supply added to a CM-grass silage-based diet, in 6 multiparous multicatheterized Holstein cows. Using a double 3 × 3 Latin square, balanced for residual effects, with 3 21-d periods, each cow was offered a fixed amount of 3 grass silage-based diets, including the following protein sources: 1) SBM (SBM_diet; 14.5% DM); 2) canola meal (CM_diet; 21.1% DM); or 3) CM_diet plus 12 g of urea/kg DM (CMU_diet) on MPY and trans-organ net fluxes of nutrients. The SBM_diet was balanced to meet MP, RDP and NEL requirements (NRC, 2001). The CM_diet was balanced to be iso-N and iso-NEL with the SBM_diet (NRC, 2001). The SBM_diet and CM_diet provided sufficient RDP whereas the CMU_diet supplied a large excess of RDP. On the last 4 d of each period, DMI and milk production and composition were determined. On the last 3 d (2 cows per d), 6 blood samples were collected from arterial, portal, hepatic and mammary vessels plus 3 spot samples of feces and urine. Data were analyzed using the Mixed procedure of SAS, and pre-planned contrasts were used to compare CM_diet to SBM_diet and CM_diet to CMU_diet. Despite lower estimated MP supply with CM_diet vs. SBM_diet (2591 vs. 2779 g/d), milk true protein yield tended to be higher in CM_diet than in SBM_diet. The CM_diet also tended to increase the efficiency of N utilization and to decrease the proportion of urinary urea-N relative to total N compared with SBM_diet. Of the EAA, only Met arterial concentration tended to increase with CM_diet compared with SBM_diet; however trans-organ net fluxes across the splanchnic tissues and the mammary gland were not affected. The net portal appearance of propionate tended to be greater in CM_diet than in SBM_diet. None of the net flux measurements supports the lower NRC (2001) predictions of MP and energy supply when CM substitutes SBM, indicating that CM is an adequate protein source in dairy ration. On the other hand, excess RDP supply decreased the efficiency of N utilization, increased plasma urea-N concentration, urinary urea-N excretion, in agreement with increased net portal absorption of ammonia, and hepatic and splanchnic release of urea-N. Although excess of RDP increased hepatic removal of ammonia, it did not affect hepatic removal of EAA and therefore, did not negatively impact milk and MPY. Therefore, although RDP supply was progressively increased to be 40% higher than recommended, this level of excess supply had no effect on net liver removal and TSP net flux of EAA, so that elevated rumen-derived ammonia production incurs no penalty on EAA availability and animal performance.

PMID 42285490
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PubMedMikrochimica acta2026-06-13

Interlaced 2D cellulose networks with molecular enrichment capability for sensitive SERS detection of sweat biomarkers.

Lin Luyao L, Wang Haonan H, Lei Xinlin X, Zhuang Xin X et al.

Efficient localization of analytes near plasmonic hotspots remains a major challenge for surface-enhanced Raman scattering (SERS) detection in complex liquid-phase systems. Herein, an interlaced cellulose-based porous membrane composed of dissolving pulp fibers (DPFs), mechanically ground nanofibers (MGNFs), sodium alginate (SA), and Ag nanoparticles was developed as a molecular enrichment-assisted SERS platform for sweat biomarker determination. The hierarchical porous architecture provided interconnected transport channels and abundant interfacial adsorption sites, facilitating analyte retention and localized enrichment within the plasmonic region. Benefiting from the synergistic effects of porous confinement and uniformly distributed Ag nanoparticles, the optimized substrate exhibited sensitive and reproducible SERS performance with an enhancement factor of 4.36 × 10⁷, a relative standard deviation of 8.04%, and a detection limit down to 1.0 × 10⁻⁸ mol/L for Rhodamine 6G (R6G). Systematic adsorption experiments using molecules with different charge properties further demonstrated the broad molecular enrichment capability of the structured cellulose network. The developed platform enabled quantitative detection of lactate and urea within physiologically relevant sweat concentration ranges and showed satisfactory analytical performance in spiked sweat samples. More importantly, this work demonstrates a structure-engineered porous membrane strategy for integrating molecular enrichment with plasmonic sensing, providing new insight into cellulose-based SERS platforms for complex bioanalytical applications.

PMID 42286362
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PubMedBMC neurology2026-06-13

Identification of signal-based gait features and blood analytes associated with stroke status and walking speed in mild acute ischemic stroke.

Şahin Erdoğan Meryem M, Özgün Mete M, Kaya Dilaver D, Akanyeti Otar O et al.

Assessment of mild acute ischemic stroke (mAIS) can be difficult, especially in regions where access to neuroimaging is limited. Integrating routine blood analyses with wearable gait assessments may aid in the identification of mAIS and estimation of functional outcomes. In this pilot study, we focus on identifying candidate gait and blood analytes associated with stroke status and functional outcomes in mAIS. Video, smartphone, and blood data were collected from 22 mAIS patients and nine healthy controls. Ridge-penalized logistic regression nomograms were developed; one to estimate the stroke status using gait, and a second one to estimate walking speed of patients using blood analytes. Our gait-based nomogram identified mAIS with an area under the curve (AUC) of 0.878, while blood-based nomogram estimated walking speed with an AUC of 0.906 (both optimism-corrected). Identified gait features for stroke status included lower xgyr_energy, xgyr_max, xgyr_std, zgyr_energy and zacc_rms, and higher zgyr_iqr, while higher age, blood urea nitrogen (BUN), and lower estimated glomerular filtration rate (eGFR) and mean corpuscular hemoglobin concentration (MCHC) were associated with slower walking. We show the feasibility of integrating gait statistics with blood analytes to identify mAIS and estimate walking speed. The nomograms showed strong discrimination and calibration within our small cohort. These findings point to the potential of multimodal signal-based features in stroke detection and rehabilitation planning, particularly in low-resource settings.

PMID 42286488
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PubMedTranslational research : the journal of laboratory and clinical medicine2026-06-13

A novel spontaneous rat model of chronic kidney disease with mitochondrial dysfunction driven by thioredoxin insufficiency.

Ohmori Iori K IK, Ouchida Mamoru M, Hada Yoshiko Y, Uchida Haruhito A HA et al.

Chronic kidney disease (CKD) is a global health burden with high prevalence and poor prognosis. Although oxidative stress and mitochondrial dysfunction have been implicated in its pathogenesis, in vivo causal evidence remains limited. Thioredoxin (Trx), encoded by Txn1, is a redox-active protein that plays a central role in controlling oxidative stress and maintaining intracellular redox homeostasis. To address this gap, we investigated the lifelong phenotypes of Txn1-F54L mutant rats harboring approximately one-third of the normal Trx activity. These rats were generated via N-ethyl-N-nitrosourea mutagenesis and validated by clustered regularly interspaced palindromic repeat (CRISPR)/CRISPR-associated protein 9 genome editing. Comprehensive analyses included biochemical testing, histopathology, immunohistochemistry, transmission electron microscopy, RNA-sequencing, western blotting, and cytokine profiling. Txn1-F54L mutant rats spontaneously developed progressive CKD, with median survival times of 110-119 days for homozygotes and 303-346 days for heterozygotes. Their clinical features-elevated blood urea nitrogen, hypoalbuminemia, hypercholesterolemia, hypertension, and arterial medial sclerosis-closely resembled those of human CKD. Histopathological evaluation revealed extensive tubular injury, interstitial fibrosis, and glomerulosclerosis. Transcriptomic profiling identified 3,418 differentially expressed genes significantly enriched in immune activation and fibrosis pathways. Mitochondrial dysfunction was prominent in proximal tubules, accompanied by oxidative stress accumulation and concurrent activation of regulated cell death pathways (apoptosis, necroptosis, and pyroptosis). Elevated serum levels of interleukin-1β, interleukin-6, and interferon-γ indicated systemic inflammation. Our findings demonstrate that lifelong Trx deficiency induces oxidative stress-mediated mitochondrial dysfunction and regulated cell death, leading to inflammation and progressive CKD. This study establishes the Txn1 mutant rat as a valuable spontaneous CKD model, providing translational insights and a platform for developing therapeutic strategies targeting oxidative stress-induced pathways.

PMID 42285432
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PubMedScientific reports2026-06-13

Dietary lactic acid and rosemary leaf supplementation enhances growth and immune responses in Nile tilapia (Oreochromis niloticus).

Menshawy Essam E, Elazeez Eman N Abd ENA, Khattab Ibrahim M IM, Abdo Safaa E SE et al.

The present study investigated the individual and combined effects of lactic acid and rosemary meal on growth performance, biochemical parameters, immune responses, the expression of growth and antioxidant-related genes, intestinal morphology, and oxidative status in Nile tilapia (Oreochromis niloticus). A total of 120 apparently healthy fish, with an average weight of 3.03 ± 0.02 g, were randomly assigned to four equal groups, each consisting of three replicates. Four experimental diets were formulated: a basal control diet (CON), a basal diet supplemented with 1 g of lactic acid per kg of diet (LA), a basal diet containing 10 g of rosemary per kilogram of diet (RM), and a basal diet that included both supplements (LA + RM). Fish were fed these diets for a duration of 60 days. The results indicated that either lactic acid or rosemary alone or in combination had a greater growth-stimulating impact than the CON group (P ≤ 0.05) with superiority to the combination group (LA + RM group). Activities of aspartate aminotransferase and alanine aminotransferase, along with creatinine and urea levels, were significantly reduced (P ≤ 0.05) in the groups of lactic acid and rosemary alone or in combination relative to the CON group. Total protein and albumin concentrations were elevated in the LA + RM group (P ≤ 0.05). Intestinal histology revealed normal morphology across groups, with increased villus height, intestinal villi spacing, and goblet cell density in LA + RM (P ≤ 0.05) without pathological lesions in the liver and spleen. Antioxidant, immune, and growth-related gene expressions were upregulated in RM and LA + RM groups. In conclusion, rosemary supplementation, alone or combined with lactic acid, enhanced fish health status and upregulated target genes without pathological lesions with superiority to the combination treatment.

PMID 42286034
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