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tafluprost + timolol maleate (Tapucom / STN 10111 / STN 1011101)

✓ Approved

Santen Pharmaceutical Co., Ltd. · ADRB1 · 小分子

什么是 tafluprost + timolol maleate?

tafluprost + timolol maleate 是一种小分子,由Santen Pharmaceutical Co., Ltd.研发。该药已获批,用于治疗相关适应症,给药途径:Others、Topical。

药物档案

商品名Tapucom, STN 10111, STN 1011101
公司Santen Pharmaceutical Co., Ltd.
药物类别小分子
分子靶点ADRB1, ADRB2, PTGFR
给药途径Others, Topical
状态Approved

作用机制

分子靶点

tafluprost + timolol maleate 作用于 3 个分子靶点:

ADRB1adrenoceptor beta 1 (B1AR, RHR)
ADRB2adrenoceptor beta 2 (ADRBR, B2AR)
PTGFRprostaglandin F receptor (FP)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

tafluprost + timolol maleate 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Eye disordersGlaucoma✓ Approved

相关研究文献

PubMedMaterials today. Bio2026-08-02

Engineering adaptive self-healing biomaterials from jammed microfluidic elastomeric particles.

Kieda Jennifer J, Ramsay Kaitlyn K, Jiang Richard R, Landau Shira S et al.

Biomaterials designed for implantation must accommodate the dynamic mechanical and structural environment of the human body. Yet, current strategies for creating materials capable of adapting their shape post-implantation remain limited. In this work, we introduced a remoldable, biodegradable, and biocompatible granular scaffold composed of monodisperse poly(octamethylene maleate (anhydride) citrate) (POMaC) particles. Monodisperse POMaC droplets with controlled diameters were generated using a droplet microfluidic platform, then subsequently jammed and UV-crosslinked to form interconnected, porous, and self-healing elastomeric scaffolds. The scaffold chemical composition and crosslinking parameters directly influenced mechanical properties, stability, and permeability, enabling tunability across a range of tissue engineering applications. The granular scaffold exhibited autonomous self-healing, enhanced molecular diffusivity, and robust cell infiltration, while remaining moldable into prescribed geometries under both in vitro and in vivo conditions. Notably, following implantation, the granular scaffolds could be remolded in vivo 24 h post-implantation, allowing adaptation to a desired geometry while preserving structural integrity, promoting the recruitment of pro-reparative macrophages, and facilitating vascular ingrowth. Collectively, this work established a versatile strategy for designing adaptive implantable biomaterials capable of responding to the body's dynamic environment, with broad potential applications in regenerative medicine and tissue engineering.

PMID 42540479
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PubMedCase reports in ophthalmological medicine2026-07-31

Choroidal Detachment in a Patient on a CPAP Therapy.

Żurowska Emilia E, Zwolińska Emilia E, Rospond-Kubiak Iwona I

The aim of the study is to present a rare case of choroidal detachment in a patient on continuous positive airway pressure (CPAP) therapy. A 76-year-old man on CPAP therapy due to obstructive sleep apnea presented to the ocular oncology clinic with a suspicion of an intraocular tumor. He complained of tunnel vision in red, floaters and flashes in the visual field, and irritation of the left eye since 13 weeks. On initial assessment, the best corrected visual acuity (BCVA) of the left eye was 1.0, and the intraocular pressure (IOP) was 21 mmHg. The examination revealed dilated, tortuous episcleral vessels and a massive choroidal effusion. The patient was diagnosed with choroidal detachment and was treated with topical dexamethasone 0.1% and cyclopentolate. On a follow-up visit 3 weeks later, the BCVA got worse to hand movements and IOP increased to 27 mmHg. The patient received a combination of dorzolamide and timolol in addition to the aforementioned treatment. Over the following 16 weeks, a gradual resolution of the choroidal detachment was documented. The CPAP treatment is a possible, though unproven, contributor to the choroidal detachment. The patient improved during corticosteroid, cycloplegic, and IOP-lowering treatment.

PMID 42534308
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PubMedBulletin of experimental biology and medicine2026-07-28

Comparative Analysis of Novel Derivatives of Pyridoxine and Dicarboxylic Acids as Activators of Transcription Factor Nrf2.

Balakina A A AA, Podgurskaya A D AD, Amozova V I VI, Stupina T S TS et al.

We performed a structure-activity relationship analysis of novel maleic acid and pyridoxine derivatives, as well as epigid and morpholine fumarates, as potential inducers of Nrf2 transcription factor. A reduction in the number of hydroxyl groups in the structure of the compounds was shown to decrease their cytoprotective activity. The effectiveness of the compounds as Nrf2 activators depends not only on the presence of maleate or fumarate moieties, but also on the structure of the hydroxyaromatic fragment of the molecule. A derivative of pyridoxine and maleic acid, 3-hydroxy-4,5-bis(hydroxymethyl)-2-methylpyridin-1-ium hydromaleate, is an effective activator of Nrf2 transcription factor and exhibits cytoprotective and antioxidant activity in vitro, which suggests its further evaluation in in vivo models and its potential for novel drug development.

PMID 42509432
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PubMedThe Journal of organic chemistry2026-07-27

Catalytic Hydrosulfenylation of Maleic Anhydride and Its Derivatives Enabled by Proton-Coupled Electron Transfer.

Peng Dong D, Sun Jiayi J, Huang Yun Y, Zeng Xianghua X

We herein report a practical method for the efficient hydrosulfenylation of maleic anhydride and its derivatives by decavanadate-induced proton-coupled electron transfer. Preliminary mechanistic studies suggest that a thiyl radical is generated from the decavanadate polyanion and thiol through an oxidative PCET process. This method utilizes readily available thiols as a sulfur source and air as an oxidant and is capable of hydrosulfenylating a variety of maleic anhydrides and maleate esters with good diastereoselectivity.

PMID 42503765
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PubMedGels (Basel, Switzerland)2026-07-27

Construction of PEGMC Copolymerized Modified Hydrogel and Its Mechanism for Salt Retardation and Nutrient Immobilization in Dryland Soil.

Cheng Jianwei J, Xiang Rui R, Liu Jingcai J, Yang Baocun B et al.

Aiming at severe soil secondary salinization, poor water retention and insufficient salt tolerance of conventional acrylic-based modifiers in arid and semi-arid regions of China, a poly(ethylene glycol) maleate citrate (PEGMC) crosslinking monomer was synthesized through esterification, and a dual covalent-hydrogen crosslinked P(PEGMC/AA) hydrogel was fabricated via free radical copolymerization with acrylic acid (AA). The hydrogel was characterized by NMR, FTIR, SEM, TGA and elemental mapping, while its binding mechanism with saline-alkali ions was elucidated through DFT calculations and molecular dynamics simulations. Its amelioration performance was evaluated through swelling, soil water retention, desalination and pot germination experiments. The hydrogel exhibited outstanding water absorbency, salt resistance and dry-wet cycling stability, with swelling ratios of 712 g/g in deionized water and 285 g/g in 0.9% NaCl solution, and remained 200 g/g after four dry-wet cycles. It enhanced soil water retention remarkably (over 93% after 72 h). At 0.30% dosage, soil salt content declined from 7.1 g/kg to 1.3 g/kg with desalination efficiency exceeding 80%, owing to porous physical adsorption and chemical chelation toward Na+, Ca2+ and Mg2+, with a binding energy of -136.936 kJ/mol. Pot tests revealed that crop germination rate rose from 19% (blank) to 75% under severe saline-alkali stress. Meanwhile, the hydrogel inhibited nutrient leaching and favored soil-water conservation. This work first incorporated PEGMC monomer into agricultural hydrogels to construct a stable dual crosslinked network, clarifying its synergistic mechanisms for salt fixation and water retention macroscopically and microscopically. It provides a promising functional material and theoretical basis for green, efficient in situ amelioration of dryland saline-alkali soil.

PMID 42505278
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PubMedFASEB journal : official publication of the Federation of American Societies for Experimental Biology2026-07-25

Syringaresinol Attenuates Aging-Associated Ferroptosis-Relevant Stress Through an HIF-1α-GPX4 Defense Axis.

Li Ya-Ping YP, Huang Fei-Hong FH, Wu Meng-Ting MT, Chen Meng-Yi MY et al.

Ferroptosis contributes to aging-associated functional decline, yet compounds with robust organismal efficacy and defined upstream regulatory mechanisms remain limited. Here, we established a diethyl maleate (DEM)-induced glutathione depletion model in wild-type (N2) Caenorhabditis elegans as a survival-based screening platform and identified syringaresinol (Syr) as a leading hit from an in-house small-molecule library. In nematodes, Syr improved survival under DEM challenge, reduced lipid peroxidation, reactive oxygen species (ROS), and malondialdehyde levels, and alleviated age-associated oxidative lipid stress and iron imbalance during natural aging, accompanied by extended lifespan and improved healthspan-related phenotypes. In primary human foreskin fibroblasts, Syr conferred dose-dependent protection against RSL3- or erastin-induced ferroptosis, preserved cellular integrity, suppressed lipid peroxidation and ROS, and restored expression of GPX4, SLC7A11, and ferritin. In two senescence models, Syr also attenuated senescence-associated phenotypes and ferroptosis-related oxidative lipid stress, concomitant with recovery of GPX4 expression. Network-based prediction and functional perturbation identified HIF-1α as a candidate mediator of Syr-associated cytoprotection. HIF-1α knockdown weakened Syr-mediated protection and largely prevented GPX4 restoration, whereas GPX4 knockdown did not alter HIF-1α abundance. These findings support a functional HIF-1α-GPX4 defense axis in fibroblasts, while direct transcriptional regulation remains to be clarified. Overall, Syr attenuates ferroptosis-relevant oxidative lipid stress and aging-associated phenotypes in C. elegans and human fibroblast models, supporting further mechanistic and mammalian in vivo validation.

PMID 42501322
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