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sumatriptan (Alsuma autoinjector / sumatriptan, King / Alsuma)

✓ Approved

US WorldMeds, LLC · HTR1D · 小分子

什么是 sumatriptan?

sumatriptan 是一种小分子,由US WorldMeds, LLC研发。该药已获批,用于治疗相关适应症,给药途径:Injectable (Others)、Subcutaneous Injection。

药物档案

商品名Alsuma autoinjector, sumatriptan, King, Alsuma
公司US WorldMeds, LLC
药物类别小分子
分子靶点HTR1D
给药途径Injectable (Others), Subcutaneous Injection
状态Approved

作用机制

分子靶点

sumatriptan 作用于 1 个分子靶点:

HTR1D5-hydroxytryptamine receptor 1D (HTR1DA, HT1DA)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

sumatriptan 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Nervous system disordersMigraine✓ Approved

相关研究文献

PubMedJournal of animal science2026-06-13

Ruminal archaea and bacteria metatranscriptomic responses to supplementation in steers fed low-quality forage.

Fontenot Alyson B AB, Holland Laura Z LZ, Cox Jodi R JR, Falk Taylor A TA et al.

A basal diet of low-quality forage (LQF) results in decreased forage utilization and animal performance. Protein and starch supplementation can ameliorate these effects by providing additional nitrogen and energy to ruminal microbes. However, the effect of protein and starch supplementation on ruminal microbial gene expression, specifically pathways involved in methanogenesis, is not well-documented. We aimed to evaluate the effect of supplement composition on ruminal microbial gene expression before and after supplementation in steers consuming a basal diet of LQF. Five ruminally-cannulated Angus steers (BW 375 ± 45 kg) were used in a 4 × 4 Latin square and fed a basal diet of King Ranch Bluestem Hay (3.5% CP, 73% NDF), and one of four isonitrogenous (130 mg nitrogen/kg BW) supplements. Ruminal samples collected from the steers provided the two most divergent supplements, 2% starch (43% CP; 100% soybean meal) and 56% starch (21% CP; 78% corn, 19% soybean meal, 2.4% urea) were used for metatranscriptomic analysis. Samples were collected via cannula prior to and 4h post-supplementation; total RNA was sequenced. Differentially expressed genes (DEG) were identified and functionally annotated; pathway enrichment analysis was completed. Sampling time exerted a greater effect than starch concentration (∼78 vs. 17% in both archaea and bacteria). All methanogenesis pathways were differentially regulated by time (P < 0.05) with upregulated genes primarily expressed by Thermoplasmata and downregulated genes primarily expressed by Methanobrevibacter. Acetoclastic and methylotrophic methanogenesis pathways were differentially regulated by starch supplementation (P < 0.05) with upregulated genes primarily expressed by Thermoplasmatales and downregulated genes primarily expressed by Methanomethylophilus alvus. The majority of bacterial DEG were expressed by Clostridia, but unclassified Bacteroidetes was the predominant bacteria responsible for expression of carbohydrate active enzymes (CAZymes). Time relative to feeding, rather than starch supplementation, resulted in a greater number of bacterial CAZymes expressed. Supplement composition elicited changes in the taxa involved in methanogenesis and carbohydrate metabolism, suggesting the potential for effects on CH4 emissions. Further research is needed to directly quantify CH4 emissions in response to supplementation to potentially optimize supplementation strategies and improve sustainability of beef cattle production.

PMID 42286418
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PubMedBMC plant biology2026-06-12

Genome-wide identification of WRKY gene family reveals its regulatory role in ABA/CBF-mediated cold adaptation in king grass (Pennisetum purpureum × P. americanum).

Lai Xianjun X, Xiao Qimeng Q, Chen Zihan Z, Liu Siqi S et al.

King grass is a fast-growing C4 perennial with high biomass potential, yet its productivity is limited by cold stress. WRKY transcription factors (TFs) regulate abiotic stress responses, but their roles in king grass cold adaptation remain unclear. WRKY TFs were identified genome-wide using BLASTP and HMMER, followed by phylogenetic classification, transcriptome profiling, promoter cis-element analysis, weighted gene co-expression network analysis (WGCNA), molecular docking, and yeast heterologous expression assays. Sixty-two PsiWRKY genes were identified and classified into three groups. Time-series transcriptome analysis across nine cold-stress time points revealed four expression patterns, with 29 genes significantly induced (> 2-fold), mainly during late acclimation (48-72 h). qRT-PCR confirmed RNA-seq trends (R² = 0.742). Functional enrichment and WGCNA analyses indicated that cold-responsive PsiWRKYs coordinate abscisic acid-gibberellin antagonism and sugar metabolism. Molecular docking predicted interactions between PsiWRKY proteins and Calvin cycle enzymes, with PsiWRKY16 and PsiWRKY55 showing the highest structural confidence (pTM > 0.75). Network analysis identified PsiWRKY16 and PsiWRKY50 as hub regulators linking GA signaling genes (GID1/DELLA) with sugar metabolism enzymes such as GAPDH and PRK. Yeast assays quantitatively confirmed enhanced cold tolerance, as heterologous expression of PsiWRKY16 reduced doubling time by 0.56 h and increased area under the curve and carrying capacity by 26.20 and 3.39, respectively, while PsiWRKY50 increased these values by 14.45 and 1.43. Promoter analysis showed enrichment of ABRE and DRE elements (p = 0.00061), and integrative target prediction identified 193 genes co-regulated by WRKY and CBF pathways, supporting ABA-CBF signaling convergence. PsiWRKYs exhibit subgroup-specific and time-resolved responses to cold stress. PsiWRKY16, PsiWRKY50, and PsiWRKY55 are implicated in coordinating hormonal signaling and metabolic reprogramming, providing candidate targets for cold-tolerant breeding in king grass.

PMID 42277708
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PubMedNew microbes and new infections2026-06-12

Prevalence of Transfusion-Transmitted Viruses Among Blood Donors at King Fahad Armed Forces Hospital, Jeddah, Saudi Arabia (2019-2024).

Sindi Nariman N, Alzahrani Osama A OA, Alamoudi Lamis M LM, Sait Ahmad M AM et al.

To assess the prevalence, temporal trends, and diagnostic concordance of transfusion-transmitted viruses (TTVs) using combined serological and nucleic acid testing (NAT) in a large donor population in Jeddah, Saudi Arabia. This retrospective study analysed all blood donations screened from 2019 to 2024 at King Fahad Armed Forces Hospital, using serological assays and NAT. Prevalence estimates were calculated with 95% confidence intervals. Temporal trends were evaluated using generalised estimating equations logistic regression. Multivariable logistic regression identified predictors of Hepatitis B Virus (HBV) and Hepatitis C Virus (HCV) positivity. Diagnostic agreement between serology and NAT was assessed using Cohen's kappa statistic. Among 48,151 donors, seroprevalence was 0.4% for HBsAg, 0.3% for HCV Ab, 0.1% for HIV Ab, and 0.02% for HTLV Ab. HBc Ab was detected in 4.7%. NAT identified HBV and HCV in 0.2% and 0.1%, respectively. Logistic regression showed a significant annual decline in HBsAg and NAT-HBV. Older age and non-Saudi nationality were linked to higher HBsAg and HCV positivity. Concordance between serology and NAT was substantial for HIV but negligible for HBV and HCV. TTVs rates are low and declining, but HBV/HCV concordance underscores the need for continued dual testing to ensure transfusion safety.

PMID 42282993
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PubMedBasic & clinical pharmacology & toxicology2026-06-12

Targeting AVEN Liquid-Liquid Phase Separation in Colorectal Cancer: Insights From a Raddeanin A-Based Chemical Probe.

Yu Xichao X, Wu Hui H, Guo Kezhen K, Liu Zihao Z et al.

Mitochondrial dysfunction is a pivotal pathogenic mechanism in colorectal cancer (CRC), which is further exacerbated by dysregulated liquid-liquid phase separation (LLPS). However, the mechanisms underlying mitochondrial dysfunction and LLPS, as well as their therapeutic targeting, remain unclear. Using Raddeanin A as a probe and through multiomics analysis, we identified apoptosis and caspase activation inhibitor (AVEN) as a potential therapeutic target. AVEN was significantly upregulated in CRC tissues and localized near mitochondria-endoplasmic reticulum contact sites (MERCS). Biophysical assays confirmed that AVEN undergoes LLPS via its intrinsically disordered regions (IDRs). Critically, we found that AVEN IDRs orchestrate mitochondrial homeostasis through dual LLPS-dependent mechanisms: inhibiting apoptosis and facilitating post-damage mitochondrial transfer. Furthermore, we identified sumatriptan (SUM) as a potent inhibitor of AVEN IDRs, which demonstrated promising therapeutic efficacy in mouse models and clinical cohorts. Our study highlights the critical role of AVEN in regulating mitochondrial homeostasis via LLPS and suggests that targeting AVEN represents a promising therapeutic strategy for CRC.

PMID 42281486
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PubMedJournal of professional nursing : official journal of the American Association of Colleges of Nursing2026-06-12

Reclaiming nursing's power: Advancing national leadership through the revival of nursing theory.

Friend Mary Louanne ML

The United States faces persistent health inequities, chronic disease, and escalating mental health and social crises. As members of the largest and most trusted health profession, nurses are well positioned to contribute to national health leadership. Yet recent emphases on competencies, outcomes, and interprofessional training have sometimes reduced attention to the theoretical preparation needed for leadership and governance. This article argues that renewed, critical engagement with nursing theory can strengthen nurses' preparation for leadership and policy roles and outlines implications for nursing education, leadership, practice, and research. This article reviews nursing theory, acknowledging critiques of grand theories and the field's movement toward more pluralistic, empirically grounded, and equity-focused frameworks. It illustrates how Watson, Newman, and King can inform leadership and governance when used critically and alongside contemporary critical and decolonial perspectives. Educational strategies are proposed to connect theory with policy and leadership content, including mapping theories across curricula, embedding political and economic literacy, and developing longitudinal leadership pathways. Nursing has made progress in policy and leadership education, yet nurses remain. underrepresented in governance relative to their potential influence. Reclaiming nursing theory as a living, evolving resource can enhance conceptual, ethical, and systems-level thinking.

PMID 42276640
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PubMedBMJ open2026-06-12

Lived experiences, challenges and coping strategies of patients with spinal cord injury using intermittent catheterisation in Riyadh, Saudi Arabia: a qualitative study.

Abuzied Yacoub Y, Al-Amer Rasmieh R, Abdul Halain Azura A, Japar Salimah S

This study explored the lived experiences, challenges and coping strategies of Arab male patients with spinal cord injury (SCI) who rely on intermittent catheterisation (IC) to manage neurogenic bladder. A descriptive qualitative approach was employed, with data analysed using a phenomenological framework. Rehabilitation Hospital, King Fahad Medical City, Riyadh, Saudi Arabia. Male patients with SCI undergoing rehabilitation and performing IC were included in the study. Although both male and female patients were approached to participate, all eligible female patients declined participation. During the recruitment process, some female patients informally expressed privacy concerns and discomfort related to discussing bladder management issues and genital care, which may have contributed to their decision to decline participation. 10 male participants with SCI were recruited after eligible female patients declined participation. Three main themes, each with associated subthemes, emerged to reflect the participants' experiences. Theme 1: Frequent use of IC in daily life, comprised four subthemes: (1) frequency of practice, (2) environmental and health-related challenges, (3) privacy during IC and (4) fluid intake and output. Theme 2: Cleanliness and general care included two subthemes: (1) catheter cleaning and (2) incontinence. Theme 3 focused on body image and sexuality. Cultural and social norms, including privacy concerns and sensitivities surrounding intimate care in the local context, played a significant role in shaping participants' experiences and coping strategies. IC was associated with challenges affecting multiple aspects of daily life among patients with SCI, including social interactions and body image. Participants described various coping strategies used to manage the physical and psychological demands associated with IC. These experiences appeared to be influenced by cultural considerations, including privacy, modesty and sensitivity surrounding urinary care within the local Saudi context.

PMID 42276795
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