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streptokinase (Heberkinase)

✓ Approved

YM BioSciences Inc. · PLG · 重组蛋白

什么是 streptokinase?

streptokinase 是一种重组蛋白,由YM BioSciences Inc.研发。该药已获批,用于治疗相关适应症,给药途径:Injectable (Others)、Intravenous (IV)。

药物档案

商品名Heberkinase
公司YM BioSciences Inc.
药物类别重组蛋白
分子靶点PLG
给药途径Injectable (Others), Intravenous (IV)
状态Approved

作用机制

分子靶点

streptokinase 作用于 1 个分子靶点:

PLGplasminogen (HAE4)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

streptokinase 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Cardiac disordersMyocardial infarction✓ Approved

相关研究文献

PubMedArchives of microbiology2026-06-06

Mechanisms underlying pyogenic bacterial infections of the skin.

Huang Can C, Yan Xueqin X, Xu Xiangxiang X, Yang Yaru Y et al.

Pyogenic skin infections are commonly caused by Staphylococcus aureus (SA), Streptococcus pyogenes (GAS), and Pseudomonas aeruginosa (PA). Although these pathogens differ markedly in phylogeny, cell structure, and ecological adaptation, they converge on a coordinated pathogenic cascade encompassing adhesion, invasion, immune evasion, remodeling of the suppurative microenvironment, and nutrient acquisition. This review systematically compares the common pathological mechanisms underlying SA, GAS, and PA, while also delineating pathogen-specific virulence strategies of SA, GAS, and PA across key stages of infection, with representative molecular determinants including surface adhesins and coagulase in SA, M protein and streptokinase in GAS, and type IV pili and the Psl exopolysaccharide in PA. Particular focus is placed on how these bacteria evade complement- and phagocyte-mediated clearance, disrupt neutrophil function, remodel neutrophil extracellular traps (NETs) dynamics, alter coagulation-fibrinolysis balance, adapt to hypoxic lesions, and compete for restricted host nutrients. Although the three pathogens converge on pyogenic lesion formation as a shared pathological endpoint, they elicit distinct histopathological and clinical lesion phenotypes, including localized abscesses, rapidly progressive necrotizing soft-tissue infections, and chronic non-healing exudative wounds. These similarities and differences indicate that suppuration is not merely the endpoint of inflammation, but a dynamic pathogenic microenvironment jointly shaped by bacterial virulence and host responses. A clearer understanding of these common pathological axes and pathogen-specific differences provides a theoretical basis and new perspectives for the development of antibacterial and host-directed therapeutic strategies in pyogenic skin infections.

PMID 42249917
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PubMedJACC. Case reports2026-06-03

4D TEE-Guided Thrombolysis for Mechanical Mitral Valve Obstruction.

Tulsidas Gitte Pramod P, Khedkar Umesh U, Kharche Milind M

To describe, step by step, how 4-dimensional transesophageal echocardiography (4D TEE) can differentiate thrombus-predominant mechanical mitral valve obstruction from pannus and thereby guide urgent thrombolytic therapy. A 24-year-old man with a 25-mm mechanical mitral prosthesis presented with NYHA functional class III dyspnea, pulmonary congestion, and a subtherapeutic international normalized ratio of 1.2. Transthoracic echocardiography showed markedly elevated transmitral gradients, and cine-fluoroscopy demonstrated restricted single-leaflet motion. TEE confirmed prosthetic obstruction, whereas 4D TEE provided the decisive mechanistic information by showing a large mobile thrombus with coexisting left ventricular-side pannus, indicating thrombus-predominant obstruction. Streptokinase thrombolysis restored bileaflet mobility and reduced transprosthetic gradients markedly. Elevated prosthetic gradients and restricted leaflet motion confirm obstruction but do not reliably distinguish thrombus from pannus. Mixed pathology may be missed if multimodality imaging is not performed. In mechanical mitral valve obstruction, 4D TEE can define the dominant mechanism of obstruction, guide selection of thrombolysis vs surgery, and document treatment success.

PMID 42233911
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PubMedCureus2026-05-28

A Non-randomized Clinical Trial on the Effectiveness and Complications of Two Different Streptokinase Dosages in Elderly Patients With ST-Elevation Myocardial Infarction (STEMI).

Chandra Subhash S, Rai Prachi Jain PJ, Singh Nouratan N, Shivhare Aaditya A

Streptokinase is widely used for thrombolysis in acute myocardial infarction (AMI), but concerns about complications have led to its underutilization in elderly patients. This study aimed to compare the efficacy and safety of standard-dose, i.e., 15 lakh international units (IU), versus half-dose (7.5 lakh IU) streptokinase in elderly patients with ST-elevation myocardial infarction (STEMI). This prospective, observational study included 103 patients with STEMI aged over 70 years, admitted within 12 hours of symptom onset. Patients were divided into two groups receiving either 15 lakh IU (n = 59) or 7.5 lakh IU (n = 44) of streptokinase. Efficacy was assessed by ST-segment resolution ≥ 50% after 90 minutes. Complications and mortality were monitored in both groups. Baseline demographic and clinical characteristics were comparable between the groups. Improvement in left ventricular ejection fraction (LVEF) from admission to one month was similar (2.75% vs. 2.84%, p = 0.885), and rates of reperfusion success (78.0% vs. 77.3%) and ST-segment resolution ≥ 50% (61.0% vs. 59.1%) did not differ significantly. Complications were more frequent in the 7.5 lakh IU group, particularly major bleeding (11.4% vs. 3.4%), though differences were not statistically significant. In-hospital mortality was low and comparable between the two groups (5.1% vs. 6.8%, p = 0.690). Half-dose streptokinase demonstrated comparable efficacy to the standard dose in achieving myocardial reperfusion in elderly patients having STEMI.

PMID 42205639
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PubMedJournal of the American Society for Mass Spectrometry2026-05-01

Metabolomic Characterization of Streptococcus dysgalactiae subsp. equisimilis: Different Metabolic States in Planktonic and Biofilm Forms and the Influence of Streptokinase.

Rockstroh Jan J, Pagel Anna-Johanna AJ, Neufend Janine V JV, Siemens Nikolai N et al.

Despite the extensive research that has been conducted into the metabolism of Gram-positive bacteria, relatively little is known about the adaptations of Streptococcus dysgalactiae subsp. equisimilis (SDSE) during biofilm maturation. This study uses targeted metabolomics and MALDI MS imaging to investigate time-dependent changes in the metabolome composition. Key metabolites of energy metabolism were quantified in planktonic and biofilm bacteria. A distinct decline in the abundance of metabolites from all analyzed metabolic pathways was observed in sessile SDSE. Furthermore, we observed a broad decrease of nutrient utilization in biofilm-associated bacteria. Additionally, we examined the impact of deleting streptokinase on SDSE metabolism. Especially, concentrations of glycolysis intermediates and adenosine phosphates exhibited significant alterations when comparing the S118 strain with its mutant. The absence of the ska gene led to drastic changes in both energy and structural metabolism. These findings provide new insight into the metabolic adaptations of SDSE and represent an initial step toward understanding its role in pathogenesis.

PMID 42062893
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PubMedIndian pediatrics2026-04-27

Clinical Practices for Management of Empyema Thoracis in Children: A Survey of Pediatricians in India.

Mathew Joseph L JL, Chandrasekaran Venkatesh V, Kumar Ketan K, Kaur Satnam S et al.

This survey was conducted to explore the current status of empyema thoracis management practices of pediatricians in India, as a prelude to developing evidence-based guidelines for managing empyema. A questionnaire examining various aspects of empyema management (diagnosis, investigations, treatment, monitoring and follow-up) was prepared, refined, and pilot-tested. It was disseminated to pediatricians across the country, through a Google form link, using email and a social media platform. Responses were collated, analyzed, and presented with descriptive statistics. Ninety-four complete responses were received, mostly from pediatricians in teaching/ tertiary-care hospitals. There were significant variations in all aspects of empyema management. There was overuse of computed tomography (CT) scan (27%) and pleural fluid Cartridge Based Nucleic Acid Amplification Test (CBNAAT) (61%) in children with pleural effusion. Whilst > 80% pediatricians used ceftriaxone empirically for pneumonia and empyema, co-amoxiclav (18%), vancomycin (56%), and teicoplanin or linezolid (16%) were also used for empyema. Less than three quarters of respondents used intercostal drainage appropriately. 25% pediatricians routinely used intrapleural fibrinolytic therapy (most often streptokinase); 37% did not use it at all. The common indications were septations/loculations on ultrasonography (57%), thick pus (38%), and persisting clinical features (33%). The duration of antibiotics ranged from < 4 weeks (18%), 4-6 weeks (59%), and > 6 weeks (15%). The indications for surgical referral also varied widely, as did monitoring during therapy, and post-treatment follow-up protocols. There are significant variations in all facets of empyema management amongst pediatricians working in diverse Indian healthcare settings, underscoring the need for evidence-based guideline recommendations.

PMID 42043772
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PubMedKathmandu University medical journal (KUMJ)2026-04-24

Reversing AV Block and Cardiogenic Shock in STEMI Care: A Case Report on Use of Fibrinolysis and Inotrope without PCI in Rural Nepal.

Pradhan A A, Tamrakar P P, Bhandari J J, Mahat P P

Atrioventricular block and cardiogenic shock are critical complications of inferior wall myocardial infarction with high mortality, especially in resource-limited settings lacking percutaneous coronary intervention. We report a 53-year-old male smoker presenting to a rural hospital with acute chest pain, dyspnea, and profound hemodynamic instability with electrocardiogram showing inferior wall ST-segment elevation myocardial infarction with Mobitz type I atrioventricular block. This case highlights reversal of atrioventricular block with return of hemodynamic stablility using Streptokinase and ionotropes in a rural setting. Therefore, timely fibrinolysis and inotropes in managing inferior wall myocardial infarction with atrioventricular block and cardiogenic shock in percutaneous coronary intervention -inaccessible regions and strengthening rural ST segment elevation myocardial infarction care networks is crucial.

PMID 42028780
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