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formoterol (Forair / Atimos / CHF 1531)

✓ Approved

Novartis AG · ADRB2 · 小分子

什么是 formoterol?

formoterol 是一种小分子,由Novartis AG研发。该药已获批,用于治疗相关适应症,给药途径:Inhaled、Topical。

药物档案

商品名Forair, Atimos, CHF 1531
公司Novartis AG
药物类别小分子
分子靶点ADRB2
给药途径Inhaled, Topical
状态Approved

作用机制

分子靶点

formoterol 作用于 1 个分子靶点:

ADRB2adrenoceptor beta 2 (B2AR, ARB2)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

formoterol 针对 2 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Respiratory, thoracic and mediastinal disordersAsthma✓ Approved
Respiratory, thoracic and mediastinal disordersChronic obstructive pulmonary disease✓ Approved

相关研究文献

PubMedJMIR formative research2026-06-11

Educational Intervention on Environmentally Responsible Inhaler Prescribing Among French General Practitioners: Pilot Pre-Post Study.

Lapeyre Camille C, Urena-Dores Aurélie A, Bourdin Arnaud A, Tostain Jean-Baptiste JB et al.

Climate change is expected to cause more than 250,000 deaths annually by 2050 and could increase the prevalence of asthma and chronic obstructive pulmonary disease (COPD) by up to 30%. Pressurized metered-dose inhalers (pMDIs), primarily delivering short-acting beta-2 agonists, generate 15 to 30 times more greenhouse gas emissions than dry powder or soft mist inhalers. In France, short-acting beta-2 agonist pMDIs account for 95% of reliever therapy prescriptions, despite their limited effectiveness in controlling disease symptoms. This study aimed to evaluate the preliminary educational impact of a single educational session on French general practitioners' awareness and intended prescribing of lower-carbon inhaler alternatives. We conducted a multicenter, single-group pre-post pilot study among 34 general practitioners from 10 multiprofessional health centers in Eastern Occitanie, France, between March and October 2023. Participants were recruited through convenience sampling. The intervention consisted of a one-time 25-minute face-to-face educational session on environmentally responsible inhaler prescribing, aligned with Global Initiative for Asthma (GINA) and Global Initiative for Chronic Obstructive Lung Disease guidelines. Data were collected using self-administered online questionnaires before the intervention and approximately 3 months later. The questionnaires included 2 clinical vignettes, one on asthma and one on COPD, with 3 prescribing questions each. Responses were categorized according to whether they included a pMDI. Changes in responses between baseline and follow-up were analyzed using the Fisher exact test or chi-square test, as appropriate. A total of 34 participants completed the baseline questionnaire. Responses including a pMDI decreased from 70.6% (48/68) to 4% (3/68) for reliever therapy (P<.001) and from 21.3% (29/136) to 4.4% (6/136) for maintenance therapy (P=.003). In asthma scenarios, adherence to GINA recommendations improved, with increased responses including inhaled corticosteroid-formoterol for reliever therapy (6%, 2/34 to 38%, 13/34; P=.001) and maintenance therapy (35%, 24/68 to 56%, 38/68; P=.02). No significant improvements were observed for COPD-related prescribing scenarios. The proportion of participants reporting environmental impact as a factor influencing inhaler choice increased from 3% (1/34) to 51% (18/34). Satisfaction was high, with 93% of participants reporting being very satisfied with the intervention. This pilot study suggests that a brief educational intervention may improve general practitioners' knowledge and intended prescribing of lower-carbon inhaler alternatives, particularly in asthma scenarios. However, the outcomes were based on theoretical clinical vignettes rather than real-world prescribing data, and the study was not designed to assess the safety or clinical effectiveness of changing inhaler prescriptions. Future studies should evaluate sustained changes in real-world prescribing while ensuring individualized, clinically appropriate, and safe inhaler choices.

PMID 42274163
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PubMedCOPD2026-06-09

Symptom Improvement with BDP/FF/G Fixed Triple Inhalation Powder in Moderate to Severe COPD Patients Uncontrolled with Dual Therapies: A Non-Interventional, Open-Label, Single-Arm, Prospective Study (RESPONSE Slovenia).

Harlander Matevž M, Šubic Tjaša T, Eržen Renato R, Maček Cafuta Arjana A et al.

People living with COPD are frequently inadequately treated due to underdiagnosis or misdiagnosis. The aim of this study was to evaluate the real-world performance of the beclomethasone dipropionate/formoterol fumarate/glycopyrronium (BDP/FF/G) fixed triple combination formulated in a dry powder inhaler (DPI) in improving symptoms, lung function, and adherence in moderate to severe COPD patients uncontrolled on dual therapies. We conducted a non-interventional, open-label, single-arm, multicenter, prospective study across 19 outpatient centers in Slovenia. The primary objective was to measure symptom improvement with the COPD Assessment Tool (CAT). A total of 359 patients with moderate to severe COPD (97% classified as GOLD E, frequent exacerbators) were followed for 24 weeks. There was a significant 6-point reduction in the CAT score after switching from dual therapies to BDP/FF/G inhalation powder (95% CI: -7.0 to -5.5; p < 0.0001). FEV1 increased by 110 mL (95% CI: 90-130; p < 0.0001) and FVC by 95 mL (95% CI: 65-120; p < 0.0001), reaching a statistically significant improvement of 2.5 percentage points in the FEV1/FVC quotient. The net improvement in dyspnea severity was 50.9% (95% CI 44.7%-57.2%), as assessed using the modified Medical Research Council (mMRC) Scale. Treatment adherence improved significantly after 6 months of triple therapy. In our cohort, switching uncontrolled moderate-to-severe COPD patients from dual therapy to BDP/FF/G fixed triple inhalation powder led to significant improvements in symptoms, lung function, dyspnea, sleep quality, and treatment adherence.

PMID 42262307
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PubMedMedicine2026-06-09

Adverse event mining for Breztri and Trelegy Ellipta based on the three international pharmacovigilance databases.

Wang Junyu J, Chen Kexu K, Yun Lu L, Xu Dexiang D

This study aimed to identify adverse drug reaction (ADR) risk signals associated with budesonide/glycopyrrolate/formoterol (Breztri) and fluticasone furoate/umeclidinium/vilanterol (Trelegy Ellipta) to support clinical decision-making and risk management. ADR reports related to Breztri and Trelegy Ellipta from the FDA Adverse Event Reporting System (FAERS) database, Japanese Adverse Drug Event Report (JADER) database and Canada Vigilance Adverse Reaction database (Q3 2004 to Q2 2024) were analyzed. After deduplication, reports were categorized using Medical Dictionary for Regulatory Activities (MedDRA) to obtain System Organ Class (SOC) and preferred terms (PTs). Disproportionality analysis was conducted using reporting odds ratio (ROR) and proportional reporting ratio methods. Analysis of 394 Breztri and 18,866 Trelegy Ellipta FAERS reports (predominantly consumer-submitted, U.S.-originated) identified 47 signals across 11 SOCs for Breztri (e.g., "Drug delivery system issue" ROR = 411.16, "Intentional device misuse" ROR = 410.69) and 160 signals across 15 SOCs for Trelegy (e.g., "Chronic eosinophilic rhinosinusitis" ROR = 187.65, "Foreign body in mouth" ROR = 107.67), revealing unlabeled risks like administration errors and packaging confusion. JADER data reinforced respiratory risks (Breztri: Chronic obstructive pulmonary disease (COPD) ROR = 516.8; Trelegy: gastrointestinal fungal infection ROR = 413.11) and device-independent safety signals (e.g., Trelegy urinary retention ROR = 28.81), while CVARD highlighted region-specific concerns including Trelegy-associated vasculitis (pulmonary vasculitis n = 29) and Breztri hypertension (ROR = 7.82). Cross-database convergence confirmed core anticholinergic/cardiopulmonary risks, yet divergent signals, FAERS' device errors, JADER's infection prominence, and CVARD's immunological events, underscore geographic heterogeneity in adverse reaction profiles, necessitating tailored risk management strategies for inhaler therapies. Inhalation device-related ADRs were observed, with Breztri showing higher incidence than Trelegy Ellipta, likely due to its more complex device usage. These findings highlight the need for enhanced patient education by healthcare providers to ensure proper device use in COPD treatment. Although core respiratory and anticholinergic risks are globally relevant, infection profiles, device complications, and rare immunological events exhibit significant geographic heterogeneity, necessitating tailored risk mitigation strategies aligned with regional pharmacovigilance patterns.

PMID 42260824
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PubMedIndian journal of pediatrics2026-06-08

Randomised Controlled Trial Comparing Single Maintenance and Reliever Therapy (SMART) with Inhaled Budesonide-Formoterol Combination, Versus Conventional Budesonide and Additional As-Needed Levo-Salbutamol, in Children with Persistent Bronchial Asthma: Author's Reply.

Mathew Joseph L JL

PMID 42258037
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PubMedJournal of clinical orthopaedics and trauma2026-06-08

Short term outcome of a two-staged approach for untreated radial longitudinal deficiency in children over two years of age.

Pandey Ritesh Arvind RA, Jhariya Rupendra R

Centralization of the hand over distal ulna remains the cornerstone of management for congenital radial longitudinal deficiency (CRLD). However, centralization alone presents several technical challenges. Gradual soft tissue distraction prior to centralization is usually helpful in tackling these issues. The currentstudy observed the short term outcomes of a two-staged procedure where wrist was gradually distracted with an external fixator before performing centralization. Retrospective analysis of 20 hands (14 patients) with Heikel type 3-4 CRLD managed by two-staged approach between year 2020 and 2024 was done. In first stage, gradual distraction of the wrist was performed with an external fixator. Once sufficient distraction was achieved, centralization of wrist over distal ulna was done as second stage without doing any tendon transfer across the wrist. Clinical hand-forearm angle (HFA) and radiological ulna-metacarpal angle (UMA) before and after treatment were compared to assess the amount of correction. Mean age of children was 33.1 months; mean follow-up after centralisation was 26 months (range 18-48 months). Radial deviation was corrected from 74.3° to 12.6° (correction 61.7°, p < 0.001) and volar flexion from 66.4° to 12.0° (correction 54.5°, p < 0.001). Radiological UMA correction was 64.0° (AP, p < 0.001) and 45.5° (lateral, p < 0.001). Complications included pin-tract infection (2 hands), physeal widening (1 hand), K-wire breakage (1 hand) and finger contractures (5 hands). All were managed conservatively without compromising the final outcome. A two-staged approach of gradual distraction and centralisation achieves satisfactory preliminary short term deformity correction in children with severe RLD presenting after two years. Prior distraction simplifies centralisation and obviates aggressive releases.

PMID 42254274
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PubMedMultidisciplinary respiratory medicine2026-06-05

Recupera e Respira: A sustainable pilot model for disposal of inhalers.

Siscaro Gherardo G, Mecchia Stefano S, Gigante Giovanni G, Luoni Benedetta B et al.

Recupera e Respira, a pilot project launched in the Friuli Venezia Giulia region in Italy in 2022, addresses the environmental impact of improper disposal of respiratory inhalers. When these medical devices are disposed of as regular household waste without segregation, they contribute to pollution with aluminum and plastic, and emission of residual hydrofluoroalkane (HFA). In collaboration with Federfarma, the national association representing over 19,000 private pharmacies affiliated with Italy's National Health Service, and with the support of Assinde, a company specializing in pharmaceutical returns management and the safe disposal of expired or unused medicines, Chiesi Italy suggested and implemented an institutionally approved collection and disposal system for empty inhalers. This initiative achieved a recovery rate of 24.6% over 3 years (calculated from IQVIA sell-out data referring to the Friuli Venezia Giulia region for September 2022 to June 2025), collecting over 111,000 inhalers from regional pharmacies. Proper disposal occurred at certified facilities capable of neutralizing hazardous components at high temperatures. The project highlights the role of pharmacies in educating patients and facilitating sustainable healthcare practices. An increase in recovery rates from 22.6% to 27.3% was observed in the first 2 years of project, with a sightly decrease over the third year. Overall, this study demonstrates the model's potential scalability, aligning with Chiesi's net zero goals by 2035. The study highlights how innovative waste management systems can effectively reduce the environmental burden of inhalers and foster public engagement in sustainability.

PMID 42246273
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