Drug Database
LA

lamivudine + zidovudine + abacavir (abacavir + Combivir / Combivir + abacavir / Trizivir)

✓ Approved

Shire · · 小分子

什么是 lamivudine + zidovudine + abacavir?

lamivudine + zidovudine + abacavir 是一种小分子,由Shire研发。该药已获批,用于治疗相关适应症,给药途径:Oral (PO)。

药物档案

商品名abacavir + Combivir, Combivir + abacavir, Trizivir
公司Shire
药物类别小分子
给药途径Oral (PO)
状态Approved

作用机制

分子靶点

lamivudine + zidovudine + abacavir 作用于 1 个分子靶点:

gag-pol, HIV-1 (gag-pol)
需要更深入的分析?Noah AI 可解释复杂机制并与同类药物比较。

治疗适应症

lamivudine + zidovudine + abacavir 针对 1 个适应症,涉及 1 个治疗领域。

治疗领域疾病/病症分期
Infections and infestationsAcquired immunodeficiency syndrome✓ Approved

相关研究文献

PubMedFrontiers in pharmacology2026-08-06

Drug-associated psoriasis: a pharmacovigilance study based on the FAERS database.

Yi Sha S, Liu Aimei A, Huoshen Wuda W, Xia Dengmei D et al.

Drug-induced psoriasis has been increasingly recognized, but the spectrum of potential triggering medications remains incompletely characterized. We aimed to identify the drugs potentially associated with psoriasis using a large-scale and real-world pharmacovigilance analysis. Firstly, disproportionality analyses were used to detect psoriasis-related drug signals. Furthermore, Multivariable logistic regression and Bayesian shrinkage models were applied to evaluate the consistency of the detected associations after adjustment for available demographic and reporting-related factors. Finally, stratified analyses by sex, age, and reporter type were conducted to assess signal robustness. A total of 30 drugs showed significant associations with psoriasis. These signals involved several pharmacological categories, including anti-infective agents (e.g., Abacavir, Fluconazole, Moxifloxacin, Sulfamethoxazole), anti-inflammatory and immunomodulatory drugs (e.g., Celecoxib, Tofacitinib), cardiovascular agents (e.g., Acebutolol, Telmisartan, Clonidine), neuropsychiatric drugs (e.g., Nortriptyline, Temazepam, Zopiclone, Wellbutrin), hormonal agents (e.g., Progesterone, Prometrium), and respiratory medications (e.g., Ventolin). Bayesian correction generally attenuated extreme effect estimates but confirmed the robustness of most signals. The stratified analysis also approve the above results. Our findings suggest that multiple drug classes are associated with psoriasis signals in pharmacovigilance data. These results highlight the importance of early recognition of drug-associated psoriasis and may assist clinicians in medication review and risk stratification in routine practice.

PMID 42558881
阅读全文 →
PubMedBMJ case reports2026-08-06

Diagnostic challenge of human herpesvirus 8-associated multicentric Castleman disease in a patient living with HIV disease.

Atithammarak Sasiwan S, Suwanpimolkul Gompol G

A man in his early 30s presented with a 4-month history of low-grade fever and chronic dry cough. Three months before admission, he developed persistent low-grade fever, rash and bilateral cervical lymphadenopathy. He was diagnosed with HIV infection and started on tenofovir/lamivudine/dolutegravir. Two weeks before admission, he developed right-sided pleuritic chest pain. Chest CT revealed bilateral pleural effusions and generalised lymphadenopathy involving the lower cervical, mediastinal and axillary regions. An excisional biopsy of a right lower cervical lymph node demonstrated hyaline-vascular architecture, including 'lollipop' lesions and onion-skinning of the mantle zones. Immunohistochemistry showed human herpesvirus 8 (HHV-8)-positive plasmacytoid cells within the mantle zones, without malignant features, consistent with HHV-8-associated multicentric Castleman disease (MCD). The patient continued antiretroviral therapy and received rituximab 375 mg/m² every week for four cycles. He achieved complete resolution of the pleural effusions. This case illustrates the variable clinical presentation of HHV-8-associated MCD in a patient living with HIV.

PMID 42557001
阅读全文 →
PubMedThe Indian journal of medical research2026-08-05

Pharmaco-economic profile, effectiveness, and safety of a dolutegravir based first line ART regimen among people living with HIV in South Gujarat.

Sojitra Brijeshkumar B, Patel Chetna C, Bhatt Krishnakant Niranjanbhai KN, Pandya Sajal S et al.

Background and objectives Dolutegravir (DTG)-based first line antiretroviral therapy (ART) is preferred globally due to its high efficacy, and tolerability. In India, data on evaluation of its pharmacoeconomic impact with effectiveness and safety remains limited. This study aimed to assess the pharmacoeconomic variables, effectiveness, and safety of the dolutegravir based first line ART regimen among people living with HIV (PLHIV) in south Gujarat. Methods This prospective, and observational study was conducted at an ART centre in a tertiary care hospital. Adults (≥18 yr) receiving first-line ART for ≥6 months were enrolled (n=204) following the informed consent. Pharmacoeconomic outcomes were evaluated using analysis of cost-effectiveness, cost minimisation, cost-utility, and cost-benefit. For effectiveness, CD4 count and plasma viral load (PVL) were recorded at baseline and 6 months. The safety was assessed using causality, severity, and preventability assessment of adverse drug reactions. Results Among 204 participants, 102 received TLD (tenofovir/lamivudine/dolutegravir) and 102 TLE (tenofovir/lamivudine/efavirenz). The TLD regimen demonstrated significantly better cost effectiveness (median CER 45.7 vs. 84.7; P<0.001) and lower mean annual treatment cost [INR (₹)17,074 vs. ₹19,283; P<0.001]. Quality-adjusted life years (QALY) and disability-adjusted life years (DALY) values were comparable between regimens. Both groups showed significant CD4 improvement over 6 months; inter-regimen differences were non-significant (P=0.386). Viral suppression at 6 months was higher with TLD (99% vs. 92.2%; P=0.019). Fourteen ADRs were reported for TLD group. Interpretation and conclusions Dolutegrevir-based regime demonstrated better cost effectiveness, lower annual cost, and more consistent viral load suppression, with comparable immunological recovery and a favourable safety profile, as compared to standard ART regime.

PMID 42555682
阅读全文 →
PubMedInfectious diseases (London, England)2026-08-04

Clinical and virological characteristics of hepatitis B virus genotype E infection: a case series.

Tiecco Giorgio G, De Francesco Maria Antonia MA, Zeneli Laert L, Gottardi Federica F et al.

Hepatitis B virus (HBV) genotype E, mainly found in sub-Saharan Africa, exhibits low genetic diversity, unique molecular markers and high recombination potential but remains under-studied. This study describes the clinical and virological characteristics, mutational profiles, antiviral treatment responses and phylogenetic data of patients with confirmed HBV genotype E infection in a tertiary-care centre in northern Italy. A retrospective monocentric study was conducted at ASST Spedali Civili di Brescia, Italy, from 2015 to 2023. Patients with documented HBV genotype E who underwent genotypic resistance testing (GRT) for clinical reasons were included. Direct sequencing of the S/POL region was used for genotyping and mutation analysis, interpreted via Geno2pheno [hbv] 2.0 and Stanford HBV resistance tools. Eight patients were identified, mostly male (62.5%) and of African origin (87.5%), with a median age of 38.5 years. GRT was performed in six (75%) patients because of persistent viremia despite antiviral treatment, five (83.3%) of whom were HIV/HBV coinfected with detectable HIV viral load. Lamivudine resistance mutations (L180M, M204V) were found in one (12.5%) case, tenofovir resistance-associated mutations (M267L/I) in two (25%) and immune escape mutations in three (37.5%), including T126I, D144E and G145R. Despite GRT, treatment was not modified in four (50%) patients due to poor adherence concerns. Therapy adjustments led to viral suppression in three (37.5%) cases. In our setting, HBV genotype E infections largely occurred among migrants from endemic regions. Although nucleos(t)ide analogues are effective across genotypes, suboptimal adherence may hinder viral suppression and promote resistance.

PMID 42547309
阅读全文 →
PubMedThe Journal of the Association of Physicians of India2026-08-03

Antiretroviral Therapy in India (2025): Drugs, Indications, Contraindications, Mechanisms, and Prophylaxis (PEP/PrEP).

Deshwal Rajesh R

India has made major gains in HIV control, with nationwide scale-up of antiretroviral therapy (ART), routine viral load monitoring, and simplified dolutegravir-based regimens. Yet gaps persist in differentiated service delivery, drug-resistance surveillance, and prevention implementation (PEP/PrEP). To provide a comprehensive, India-focused review of currently available antiretroviral drugs and fixed-dose combinations (FDCs), indications and contraindications for ART initiation, core mechanisms of action by class, regimen selection and monitoring, and detailed, practical guidance on HIV postexposure prophylaxis (PEP) and pre-exposure prophylaxis (PrEP), with attention to 2024-2025 updates. Narrative review of national guidance (NACO), WHO recommendations, and key implementation documents and peer-reviewed Indian literature (2018-2025), emphasizing policy-relevant updates and practical algorithms. (1) First-line ART in India is an FDC of tenofovir disoproxil fumarate/lamivudine/dolutegravir (TLD), with alternatives guided by renal, hepatic, pregnancy, TB cotreatment, and toxicity considerations. Viral load monitoring and "Treat All" remain policy cornerstones. (2) PEP: NACO's national PEP document continues to list a 28-day triple regimen with TDF + 3TC + EFV started as soon as possible (preferably ≤2 h; within 72 h). Several institutions have operationalized DTG-based PEP (TDF/3TC/DTG) in line with broader ART updates and WHO's 2024 PEP guidance favoring 3-drug regimens. (3) PrEP in India: DCGI approved TDF/FTC for PrEP; national technical guidance exists, but programmatic rollout remains uneven. Global prevention options expanded with FDA approval (June 2025) of twice-yearly injectable lenacapavir for PrEP. Indian availability will depend on future regulatory decisions and access arrangements. India's ART platform is strong and increasingly INSTI-based. Scaling PrEP, standardizing DTG-aligned PEP, fortifying viral load and resistance monitoring, and integrating long-acting prevention as it becomes available are the next priorities.

PMID 42543939
阅读全文 →
PubMedCureus2026-08-03

Dolutegravir-Associated Dyslipidemia and Atherogenic Lipid Changes Among Treatment-Naïve People Living With HIV: A 12-Month Prospective Cohort Study From Southern India.

Sebastian Savitha A SA, Devasia Cerin C, Selvam Sumithra S, Idiculla Jyothi J

Background Dolutegravir (DTG)-based antiretroviral therapy (ART) is widely used for the treatment of people living with HIV (PLHIV). As cardiovascular disease risk becomes increasingly important in the long-term management of PLHIV, understanding changes in lipid parameters following initiation of DTG-based therapy is clinically relevant. Prospective data on dyslipidemia and atherogenic lipid indices among Indian PLHIV initiating tenofovir disoproxil fumarate-lamivudine-dolutegravir (TLD) remain limited. This study aimed to evaluate changes in lipid profiles and atherogenic indices over 12 months among ART-naïve PLHIV initiating TLD. Methodology We conducted a 12-month prospective cohort study at the HIV Clinic of a tertiary teaching hospital in Bengaluru, India. A total of 70 adult ART-naïve PLHIV initiating TLD were enrolled consecutively. Participants with baseline dyslipidemia, lipid-lowering therapy, pregnancy, or lactation were excluded. Fasting lipid profile, including serum total cholesterol (TC), low-density lipoprotein cholesterol (LDL-c), high-density lipoprotein cholesterol (HDL-c), triglycerides (TG), and atherogenic indices (TC/HDL-c ratio, TG/HDL-c ratio, non-HDL cholesterol) were measured at baseline and 12 months. Body mass index (BMI), fasting blood sugar (FBS), serum alanine aminotransferase (ALT), and serum creatinine were also recorded at these time points. Enrolled participants were followed up for 12 months to determine the one-year incidence of dyslipidemia and changes in lipid parameters and atherogenic indices. Results All 70 participants completed follow-up (100% retention; median age = 33 years (interquartile range = 27-40); 74.3% male). The main finding was that 24/70 (34.29%, 95% confidence interval = 23.5-46.7) developed incident dyslipidemia at 12 months, with 17/24 (70.8%) demonstrating ≥2 concurrent lipid abnormalities. Low HDL-c (24.29%) and hypertriglyceridemia (22.86%) were most frequent. Statistically significant adverse mean changes occurred in TC (157.1 → 164.6 mg/dL; t(69) = 2.23, p = 0.029), LDL-c (95.8 → 111.1 mg/dL; t(69) = 5.15, p < 0.001), TG (131.7 → 154.7 mg/dL; Z = 3.60, p < 0.001), non-HDL-c (108.9 → 119.8 mg/dL; Z = 2.45, p = 0.014), TC/HDL-c ratio (3.37 → 4.03; Z = 2.18, p = 0.029), and TG/HDL-c ratio (2.85 → 4.04; Z = 3.05, p = 0.002). HDL-c declined non-significantly (48.2 → 44.8 mg/dL; t(69) = -1.83, p = 0.071). BMI rose +0.67 kg/m² (t(69) = 3.43, p = 0.001), serum creatinine +0.11 mg/dL (t(69) = 4.86, p < 0.001), ALT increased by 12.6 IU/L (Z = -5.97, p < 0.001), and FBS +7.6 mg/dL (t(69) = 2.00, p = 0.049), without new diabetes. Conclusions DTG-based antiretroviral therapy (TLD) was associated with a 34.29% one-year incidence of dyslipidemia in ART-naïve Indian PLHIV, with significant adverse shifts in atherogenic indices. These findings support routine lipid and metabolic surveillance and consideration of statin therapy in eligible patients as essential components of monitoring care for PLHIV on DTG-based ART.

PMID 42544255
阅读全文 →

注册免费账户还可查看另外 9996 篇文献

免费注册查看全部文献 →

了解更多lamivudine + zidovudine + abacavir